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Adenosine receptor A1 antagonist 5
CAS No. 85872-53-3
Adenosine receptor A1 antagonist 5( —— )
Catalog No. M33817 CAS No. 85872-53-3
Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 149 | Get Quote |
|
| 5MG | 228 | Get Quote |
|
| 10MG | 333 | Get Quote |
|
| 25MG | 552 | Get Quote |
|
| 50MG | 787 | Get Quote |
|
| 100MG | 1062 | Get Quote |
|
| 500MG | 2124 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameAdenosine receptor A1 antagonist 5
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NoteResearch use only, not for human use.
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Brief DescriptionAdenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.
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DescriptionNPC 200 is a potent and selective antagonist of Adenosine A1 Receptor. NPC 200 reverses NECA-induced left and right atrial depression with EC50s of 1.08 and 2.03 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayGPCR/G Protein
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TargetcAMP
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RecptorcAMP
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Research Area——
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Indication——
Chemical Information
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CAS Number85872-53-3
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Formula Weight312.37
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Molecular FormulaC17H20N4O2
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Purity>98% (HPLC)
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Solubility——
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SMILESC(CC)N1C2=C(NC(=N2)C3=CC=CC=C3)C(=O)N(CCC)C1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. P. V. Kaplita, et al. NPC 205 is a potent and selective adenosine A1, receptor antagonist: Correlation among receptor binding, biochemical, and physiological assays. , 20(4), 429–443.
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